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The National Cancer Institute is making its inventory of radiolabeled compounds available to qualified researchers. These radiolabeled drugs are available to qualified researchers from the Drug Synthesis and Chemistry Branch, DTP, DCTD, NCI.
Requests for radiolabeled compounds should be addressed to:
Dr. Prabhakar Risbood
Drug Synthesis and Chemistry Branch
National Cancer Institute
Executive Plaza North, Suite 8028
6130 Executive Boulevard, MSC 7448
Bethesda, MD 20892-7448
| Phone: | 301-435-9157 or 301-435-9159 |
| Fax: | 301-480-4817 |
Requestor must submit a brief description of the planned research and a justification of the need for the labeled material, a request should include the amount of radioactivity needed, and the required specific activity.
These requests are reviewed by an NCI committee for approval. The labeled compounds are provided free of charge to qualifying researchers. Qualifying researchers must have a valid radioactive materials license, and a copy of the license must be sent to the NCI and to the shipping contractor. Name and address of the shipping contractor will be provided upon approval.
In addition a duly signed Simple Letter of Agreement (SLA) available in html format or PDF format and Federal Express account # must be submitted along with the request. Requestor will bear the shipping.
INCOMPLETE REQUEST FORMS WILL NOT BE PROCESSED AND NOTIFICATION OF INCOMPLETENESS WILL NOT BE SENT.
Available Radiolabeled Drugs
| NSC Number | Drug Name |
|---|---|
| 755 | [8-14C]Purine-6-thiol |
| 1895 | Guanazole[14C] |
| 3051 | [formyl-14C]N-Methylformamide |
| 3088 | 4-(p-[Bis-(2-chloroethyl)amino][14C]-phenyl) butyric Acid |
| 3801 | O-[ 14C]methylhydroxylamine hydrochloride |
| 7359 | 9-b-D-Xylofuranosyl-[8-Z14C]adenine |
| 13875 | Hexamethyl[2,4,6-14C]melamine |
| 20810 | 2R,4'R,8'R-a-[5-Methyl-14C]Tocopherylquinone |
| 51143 | 2,3-Dihydro-1H(imidazo-2,3-14C)-(1,2b)-pyrazole |
| 52695 | Cyclohexylammonium N,N-bis(2-chloro-ethyl- U-14C),-N'-3-hydroxypropylphos-phorodiamidate |
| 63878 | [2-14C]Cytosine-b-D-arabinofuranoside |
| 63984 | 3'-3H-3'-Deoxyadenosine |
| 68075 | Thalicarpine[6a, 7-3H] (in benzene) |
| 68626 | 1-Acetyl-2-picolinoylhydrazine-[carbonyl-14C] |
| 71090 | Methyl 3-(4-nitrophenyl)[1- 14 C]prop-2-ynoate |
| 73754 | Fluorodopan[chloroethyl-2-14C] |
| 92188 | 1-Formylisoquinoline[1-14C]thiosemi-carbazone |
| 92339 | (6a , 11b , 16a )-6,9-diluoro-11,21-dihydroxy-16,17-(1-methyyethylidene) bis-oxy-pregnan-[1,2-3H]-1,4-diene-3,20-dione, [1,2-3H]fluocinolone acetonide |
| 94100 | 1,6-Dibromo-1,6-dideoxy-[1-14C]-D-mannitol |
| 95580 | N,N'-[3,4-3H]Hexamethylenebisacetamide |
| 98700 | [purine-3H]2',3'-Dideoxyadenosine |
| 102627 | 3,3'-Iminodipropan-1-ol di[14C]methane sulfonate hydrochloride |
| 104801 | [phenyl-U-14C]Cytembena |
| 105831 | 2-Nitro[2-14C]imidazole |
| 112907 | [2-14C]Tetrahydrouridine |
| 113496 | 5-Aminoimidazole-4[carboxamide-2-14C]- Hydrochloride |
| 118742 | [N-methyl-14C]Pentamethylmelamine Hydrochloride |
| 125973 | [3-3H]Taxol |
| 126849 | [ribose-1-14C]3-Deazauridine |
| 127755 | 3-Chloro-4-[4-[2-chloro-4(4,6-diamino-2,2- dimethyl[4,6-14C]-s-triazin-1(2H)-yl-phenyl] butyl]benzenesulfonyl fluoride Ethanesulfonate |
| 135091 | 1-(2-Chloroethyl)-3-(cis-4-methylcyclo- hexyl-1-14C)-1-nitrosourea |
| 139105 | a-[2-Chloro-4-(4,6-diamino-2,2-dimethyl- [4,6-14C]-s-triazine-1[2H]-yl)phenoxy]-N,N- dimethyl-m-toluamide Methanesulfonate |
| 139490 | 5-[14C]Methyltetrahydrohomofolic Acid Sodium Salt |
| 141537 | Anguidine[3-3H] |
| 141549 | 9-(4-Methanesulfonamido-2-methoxy-anilino)[9-14C] acridine Monohydrochloride |
| 143414 | Benzyldimethylrifampicin[38-14C] |
| 145668 | 2,2'-Anhydro-[2-14C]-1-b-D-arabino-furanosyl- cytosine Hydrochloride |
| 154890 | [14C]Coralynesulfoacetate |
| 161128 | 1-(dimethylcarbamothioylthio)-1-methyl-3-[ 14C(U)]phenylurea |
| 176319 | 6-Amino-1-methyl-4-[(1-methylpyri-dinium-4-yl) amino]phenyl]amino][14C]car-bonyl]phenyl]amino] quinolinium Dibromide |
| 182986 | [benzoquinone-U-14C]AZQ |
| 218321 | R-[8-3H]Pentostatin |
| 219733 | N,N'-[9-Acridinyl-9-[14C]-1,6-hexane-diamine |
| 221019 | [21- 3H]Wortmannin |
| 224964 | ([4,5-3H2]1,2-cyclohexanediamine-N,N')- [propanedioato-(2-)O,O']platinum (II) |
| 234714 | Aphidicolin[17- |
| 249992 | [methanesulfonyl-14C]m-AMSA |
| 253272 | N-[1-14C]Acetyl-N-(methylcarbamyloxy)-N'- methylurea |
| 262666 | 1,4-Bis(2'-chloroethyl)-1,4-diazabicyclo- [2.2.1]heptane-7-14C Dimaleate |
| 263164 | Erythro-9-(2-hydroxy-3-nonyl)adenine-[8-14C] 1.25 Hydrochloride |
| 264074 | 1,2-Ethylene-3,3'-bis(5,5-pentamethylene- hydantoin-4-14C) |
| 264880 | [triazine-4-14C]Dihydro-5-azacytidineHydrochloride |
| 267213 | [benzenesulfonyl-14C]Glyoxylic Acid, 4-Methoxybenzenesulfonyl Hydrazone |
| 278214 | [5-14C]5-(3,4-Dichlorophenyl)-2,3-dihydro-6, 7-bis-[N-i-propylcarbamoxy)methyl]-1H-pyrrolizine |
| 279836 | [anthracenedione-[14C]DHAQ |
| 281272 | 4-Amino-1-b-D-arabinofuranosyl-[6-3H]- 1,3,5-triazine-2(1H)-one |
| 281612 | 2,2’-(4-[ 14 C]formyl-3-methylphenylazanediyl)bis(ethane-2,1-diyl)dimethanesulfonate |
| 284356 | [1,3,5,7-14C]Octahydro-4,8-ethenopyrrolo- [3',4':3,4]cyclobut[1,2f]isoindole- 1,3,5,7-(2H,6H)tetrone |
| 296934 | a-1,3,5-Tris(oxiranylmethyl)-[U-14C]- 1,3,5-triazine-2,4,6-(1H,3H,5H)trione |
| 299933 | [8-3H]Thapsigargin |
| 319726 | 2-Acetylpyridine 4,4-trimethylene-[14C]- thiosemicarbazone |
| 326231 | L-[1-14C]Buthionine, R,S-sulfoximine |
| 336628 | Hexahydro-4,6-dioxy-N-phenyl-2-thioxo-5-[2-14C] pyrimidine Carboxamide |
| 338947 | 2-chloro[1,2-14C]ethyl(methylsulfonyl)- methanesulfonate |
| 339004 | Benzenesulfonamide, 4-amino-N-(5-chloro- 2-[2,3-14C]quinoxalinyl)- |
| 347512 | [pyran-2-14C]Flavone-8-acetic acid |
| 348948 | [6,7-14C]-1,5,2,4-Dioxadithiepane-2,2,4,4-tetroxide |
| 349174 | 5-(3-Aminopropyl)amino]7,10-dihydroxy- 2[2-[(2-hydroxyethyl)amino]ethyl][6,10b-14C] anthra[1,9-cd]pyrazol-6(2H)one Dihydrochloride |
| 349438 | 1-(3-Furyl)-4-hydroxy-1-[3,3,4,5,5,5-2H6]-pentanone |
| 361456 | [2- 14C]Pyrazine, 2-diazohydroxide, sodium salt |
| 363813 | D-Tetrachloro-trans-1,2-[4,5-3H2]cyclo- hexyldiamine platinum (IV) hemihydrate |
| 364837 | [4,5-3H(n)]trans-1,2-Diaminocyclohexane dichloroplatinum (II) |
| 366140 | [10b-14C]Pyrazolo[3,4,5-kl]acridine-2-(6H)- propanamine, 9-methoxy-N,N-dimethyl-5-nitro-, monomethanesulfonate |
375574 | [uracil-5-6-3H]cyclopentenyluridine | 376128 | [3H(G)]Dolastatin-10 |
| 607097 | [1-3H]7-Cyanoquinocarcinol |
| 609974 | 1H-1,2,3-Triazole-4-carboxamide, 5-amino-1- [[3,5-dichloro-4-(4-chloro[7-14C]-benzoyl) phenyl]methyl- |
| 612049 | [hypoxanthine-3H]2',3'-Dideoxyinosine |
| 614552 | [3-14C]Castanospermine |
| 614846 | [8-14C]Carbovir |
| 615985 | Isopropyl 2-chloro-5-(2-methyl-5,6-dihydro- 1,4-oxathiin-3-yl carboxamido)-[U-14C]benzoate |
| 617990 | 2-Acetylpyridine 4,4-trimethylene[14C]-semicarbazone |
| 618074 | [alanine-2,3-3H]Alanylbatracylin |
| 618121 | 2,3-Bis(3,4-dimethoxyphenyl)-3-chloro- [3-14C]propenal |
| 620107 | [amidine-14C]Pentamidine isethionate |
| 623310 | [20-3H]Prostratin |
| 624151 | [3,6-14C]-cis-4,5-Dihydroxy-1,2-dithiane-1,1-dioxide |
| 624231 | 1 11-Nitro-2-([UL-14C]phenylsulfonyl)benzene |
| 624540 | [methyl-14C]Aurintricarboxylic Acid |
| 625487 | 1-(2,6-Difluorophenyl)-[1-14C]1H, 3H-thiazolo[3,4-a]benzimidazole |
| 627505 | 9-Methoxy-2-methyl[14C]ellipticinium acetate |
| 629243 | 1-Methylethyl 2-chloro-5-[[(1-methylethoxy) -thioxomethyl]amino][7-14C]benzoate |
| 633713 | 2-(4-carboxy-4-(4-((2,4-diaminopteridin-6-yl)- methylamino)phenylamido)butylcarbamoyl)[4,5- 3 H]benzoic acid |
| 638352 | [phenylene-14C]Quinobene |
| 643812 | 3'-O-Phosphono-(Z)-[1-14C]combretastatin A4 Disodium salt |
| 645727 | 4-Chloro-3-[[(1-methylethoxy)imino]methyl]- [UL-14C]phenyl Carbamothioic Acid O-(1-Methylethyl) Ester |
| 649890 | [ 14 C]HL-275 |
| 654021 | t-Butyl-3-isopropyl-3-[(2R,3S)-2-hydroxy-3- (N-[8-3H]quinaldoyl-L-asparaginyl)amino- 4-phenylbutyl]carbazate |
| 654663 | [phenyl- 3H] Auristatin PE |
| 654705 | 4-(2,5-Dihydroxybenzylamino)[7-14C]-benzoic acid methyl ester |
| 656202 | [7-3H]7(S)-Brefeldin A |
| 672594 | L,L-2{2-[2-(1-carboxy-2-methylbutyl[14C]carbamoyl)phenyldisulfanyl][14C]benzoylamino}-3-methylpentenoic acid |
| 674495 | 2-(4-Amino-3-methylphenly)-[2-14C]-benzothiazole |
| 680410 | 4-{[(2,5-Dihydroxyphenly)methyl]amino}[carboxy-14C]benzoic acid 1-adamantyl ester |
| 684218 | 2-(Dimethylamino)-4,5-dihydro-5-methyl-1-(4-nitrophenyl)-4-(2-oxo-propyl)-[4-14C]-1H-pyrido[3,2b]-indole-3-carbonitrile |
| 686288 3H | 5-Amino-2-(4-amino-3-fluorophenyl)-6,8-diflouro-7-methyl-[3-3H]-4H-1-benzo-pyran-4-one |
| 686288 14C | 5-Amino-2-(4-amino-3-fluorophenyl)-6,8-diflouro-7-[14C]methyl-4H-1-benzo-pyran-4-one |
| 687406 | [6a,7,8,9,10,10a-14C]Indolo[2,1-b]pteridine-6,12-dione |
| 697887 | 2-[4-(7-chloro-2-quinoxalinyloxy)[3H]phenoxy]propionic acid |
| 710305 | 5-Fluoro-2-{4[(S)-2,6-diaminohexanoyl-amino]-3-methylphenyl}-[2-14C]benzothiazole |
| 720764 | N,N',N"-Tris(2-[6-3H]pyridyl methyl)-cis-1,3,5-trimethylaminocyclo-Hexane([Methyl-3H] TACHPYR) |
| 721630 | 8-O-debutanoyl-[8-3H]thapsigargin |
| 722041 | N-Geranyl-N'-(2-adamantyl)-[1-14C]ethane-1,2-Diamine (SQ109) |
| 733625 | (3-[4-N,N-bis-2-chloroethylamino]-phenyl-[1-14C]propyl)carbamic acid, 11 b-(17b-hydroxyestra-4,9(10)-diene-3-one)-hexyl-aminoethyl ester |
| 735210 | N-[(L-trans-3-carboxyoxiran-2-yl)-carbonyl]-L-leucyl-3-(p-hydroxy-phenyl)-[1-14C]ethyl-amide, sodium salt (JPM-565 sodium salt) |
| 743380 | N-(3-chlorobenzyl)-3-hydroxy[3H]methylindole |
| 749798 | Z-1-(4-hydroxyphenyl)-1-[4-(2-[3H]methylaminoethoxy]-2-phenylbutene ([N-C3H3]Endoxifen) |